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KS 176

Catalog #: 4169 Datasheet
Catalog # Availability Size / Price Qty
4169/10
4169/50
KS 176 | CAS No. 1253452-78-6 | Multidrug Transporter Inhibitors
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Description: Selective BCRP inhibitor

Chemical Name: N-[4-(2-Hydroxyethyl)phenyl]-2-[(4-nitrobenzoyl)amino]benzamide

Purity: ≥98%

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Biological Activity

KS 176 is a selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter (IC50 values are 0.59 and 1.39 μM in Pheo A and Hoechst 33342 assays respectively). Displays no inhibitory activity against P-gp or MRP1.

Technical Data

M.Wt:
405.4
Formula:
C22H19N3O5
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
1253452-78-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Specific inhibitors of the breast cancer resistance protein (BCRP).
    Pick et al.
    ChemMedChem, 2010;5:1498

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