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TCS 2510

Catalog #: 4069
2 Citations Datasheet
Catalog # Availability Size / Price Qty
4069/1
TCS 2510 | CAS No. 346673-06-1 | Prostanoid Receptor Agonists
1 Image
Description: Selective EP4 agonist

Chemical Name: (5R)-5-[(3S)-3-Hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5-yl)hexyl]-2-pyrrolidinone

Purity: ≥98%

Product Details
Citations (2)
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Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM). Displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM.

Technical Data

M.Wt:
383.49
Formula:
C21H29N5O2
Solubility:
Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml)
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
346673-06-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Discovery of a potent and selective agonist of the prostaglandin EP4 receptor.
    Billot et al.
    Bioorg.Med.Chem.Lett., 2003;130:1129

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Citations for TCS 2510

The citations listed below are publications that use Tocris products. Selected citations for TCS 2510 include:

2 Citations: Showing 1 - 2

  1. Utilizing Designed Receptors Exclusively Activated by Designer Drug Chemogenetic Tools to Identify Beneficial G Protein-Coupled Receptor Signaling for Fibrosis.
    Authors: Tzu-Ming Et al.
    J Pharmacol Exp Ther  2020;375:357-366
  2. Prostaglandin E(2) mediates proliferation and chloride secretion in ADPKD cystic renal epithelia.
    Authors: Liu Et al.
    Am J Physiol Renal Physiol  2012;303:F1425

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