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MSC 4381

Catalog #: 8008 Datasheet
Catalog # Availability Size / Price Qty
8008/10
MSC 4381 | CAS No. 2445185-57-7 | Monocarboxylate Transporter Inhibitors
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Description: Potent and selective monocarboxylate transporter 4 (MCT4) inhibitor

Chemical Name: 5-[2-[5-Chloro-2-[[(5-ethoxy-8-quinolinyl)sulfonyl]amino]phenyl]ethynyl]-4-methoxy-2-pyridinecarboxylic acid

Purity: ≥98%

Product Details
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Biological Activity Technical Data Additional Information Product Datasheets Calculators

Biological Activity

MSC 4381 is a potent and selective monocarboxylate transporter 4 (MCT4) inhibitor (IC50 = 77 nM; Ki = 11 nM). Inhibits lactate efflux in MDA-MB-231 cells (IC50 = 1 nM) and reduces viability of cells expressing high levels of MCT4.

Technical Data

M.Wt:
537.97
Formula:
C26H20ClN3O6S
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2445185-57-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the MSC 4381 probe summary on the SGC website.

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