GSK 264220A
Chemical Name: N-[2-Methyl-5-(1-piperidinylsulfonyl)-3-furanyl]-N'-phenylurea
Purity: ≥98%
Biological Activity
GSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
-
A high-throughput screen for the endothelial lipase using HDL as substrate.
Keller et al.
J.Biomol.Screen., 2008;13:468 -
Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors.
Goodman et al.
Bioorg.Med.Chem.Letts., 2009;19:27
Product Datasheets
Citation for GSK 264220A
The citations listed below are publications that use Tocris products. Selected citations for GSK 264220A include:
1 Citation: Showing 1 - 1
-
Analysis of ECs and related compounds in plasma: artifactual isomerization and ex vivo enzymatic generation of 2-MGs.
Authors: Pastor Et al.
J Lipid Res 2014;55:966
FAQs
No product specific FAQs exist for this product, however you may
View all Small Molecule FAQsReviews for GSK 264220A
There are currently no reviews for this product. Be the first to review GSK 264220A and earn rewards!
Have you used GSK 264220A?
Submit a review and receive an Amazon gift card.
$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image
