Home / Focal Adhesion Kinase Inhibitors / GSK 2256098

GSK 2256098

Catalog #: 7786 Datasheet
Catalog # Availability Size / Price Qty
7786/50
7786/10
GSK 2256098 | CAS No. 1224887-10-8 | Focal Adhesion Kinase Inhibitors
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Description: Potent focal adhesion kinase (FAK) inhibitor

Chemical Name: 2-[[5-Chloro-2-[[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino]-4-pyridinyl]amino]-N-methoxybenzamide

Purity: ≥98%

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Biological Activity

GSK 2256098 is a potent, reversible and ATP-competitive focal adhesion kinase (FAK) inhibitor (IC50 values are 8.5 nM, 12 nM and 15 nM in U87MG, A549 and OVCAR8 cell lines respectively). Inhibits Y397 phosphorylation and motility, growth and survival of pancreatic ductal adenocarcinoma cells.

Technical Data

M.Wt:
414.89
Formula:
C20H23ClN6O2
Solubility:
Soluble to 100 mM in DMSO and to 50 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1224887-10-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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