BQ-3020
Purity: ≥95%
Biological Activity
BQ-3020 is a highly potent and selective ETB endothelin receptor agonist (Ki values are 0.18 and 970 nM at human ETB and ETA receptors respectively).Technical Data
(Modifications: Leu-1 = N-terminal Ac)
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
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Effects of selective ETB-receptor stimulation on arterial, venous and capillary functions in cat skeletal muscle.
Ekelund et al.
Br.J.Pharmacol., 1994;112:887 -
[3H]-BQ-123, a highly specific and reversible radioligand for the endothelin ETA receptor subtype.
Ihara et al.
Eur.J.Pharmacol., 1995;274:1 -
Distinct subdomains of human endothelin receptors determine their selectivity to endothelinA-selective antagonist and endothelinB-selective agonists.
Sakamoto et al.
J.Biol.Chem., 1993;268:8547 -
Pharmacological differences between rat and human endothelin B receptors.
Reynolds et al.
Biochem.Biophys.Res.Commun., 1995;209:506
Product Datasheets
Citation for BQ-3020
The citations listed below are publications that use Tocris products. Selected citations for BQ-3020 include:
1 Citation: Showing 1 - 1
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Inflammatory mediators alter the astrocyte transcriptome and calcium signaling elicited by multiple G-protein-coupled receptors.
Authors: Hamby Et al.
Cell Death Dis 2012;32:14489
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