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BAY 6096

Catalog #: 8006 Datasheet
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8006/10
BAY 6096 | CAS No. 2313483-41-7 | Adrenergic alpha-2 Receptor Antagonists
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Description: Potent and selective adrenergic α2B antagonist

Chemical Name: 1-[2-[[[3-(3,5-Dimethyl-4-isoxazolyl)imidazo[1,2-a]pyridin-7-yl]carbonyl]amino]ethyl]-4-(methylamino)pyridinium chloride

Purity: ≥98%

Product Details
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Biological Activity

BAY 6096 is a potent (IC50 = 14 nM), and selective adrenergic α2B receptor antagonist that displays 394, 725, >845-fold selectivity over α1A, α2A, and α2C, respectively. BAY 6096 reduces α2B receptor agonist-induced vasoconstriction and has a high clearance and low mean residence times in rats. BAY 6096 is highly water-soluble.

Technical Data

M.Wt:
426.91
Formula:
C21H23ClN6O2
Solubility:
Soluble to 100 mM in water and to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2313483-41-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This compound is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the BAY 6096 probe summary on the SGC website.

Product Datasheets

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